Design and synthesis of 4,5,6,7-tetrahydro-1H-1,2-diazepin-7-one derivatives as a new series of Phosphodiesterase 4 (PDE4) inhibitors

The aim of this poster is to provide a new chemical starting point to seed future drug discovery efforts. Despite the 5500 compounds already synthesized by both companies and academia, is it still possible to design a novel PDE4 inhibitor series?

Recently presented by our expert, Sara Guariento, at EFMC 2017, download your copy of our educational scientific poster today and discover more about PDE4 inhibitors.