Aptuit | Hit to lead

Hit to Lead

Converting initial Hits into drug-like NCEs

Our flexible range of strategies are proven to deliver successful and effective drug discovery projectOur Hit to Lead capabilities integrate Computational and Medicinal Chemists, DMPK, Pharmacology and Analytical Sciences expertsFollowing the identification of Hit series we work closely with you to establish which Hits should be prioritized.

Our Hit to Lead capabilities integrate Computational and Medicinal Chemists, DMPK, Pharmacology and Analytical Sciences experts. Hits are filtered based on workable chemical structures and physicochemical properties.

Focused libraries are generated around the most promising Hits for early and rapid generation of structure activity relationship data.

You can take advantage of our areas of expertise to support standalone or integrated Hit to Lead programs.